Items where authors include "Harrity, J.P.A."
Article
Hoteite, L., Allen, B.D.W., Elhajj, E.A. et al. (2 more authors) (2024) A Pd‐catalyzed annulation strategy to linearly fused functionalized N‐heterocycles. Chemistry – A European Journal, 30 (21). e202400116. ISSN 0947-6539
Han, J., Gao, W. and Harrity, J.P.A. orcid.org/0000-0001-5038-5699 (2024) Pd-Catalyzed [4 + 1] annulation strategy to functionalized 4-methyleneproline derivatives. The Journal of Organic Chemistry, 89 (3). pp. 1552-1555. ISSN 0022-3263
Gao, W., Han, J., Greaves, S. et al. (1 more author) (2023) Asymmetric synthesis of functionalizable type II β-turn-inducing α-amino acid building blocks. Organic Letters, 25 (35). pp. 6555-6559. ISSN 1523-7060
Valdez Pérez, L.F., Bachollet, S.P.J.T., Orlov, N.V. et al. (2 more authors) (2023) A dynamic thermodynamic resolution strategy for the stereocontrolled synthesis of streptonigrin. Angewandte Chemie International Edition, 62 (5). e202213692. ISSN 1433-7851
Han, J., Hoteite, L. and Harrity, J.P.A. orcid.org/0000-0001-5038-5699 (2022) Development of an enantioselective allylic alkylation of acyclic α-fluoro-β-ketoesters for the asymmetric synthesis of 3-fluoropiperidines. Chemistry – A European Journal, 28 (56). e202201595. ISSN 0947-6539
Cousins, D.L., Lim, Y.H. and Harrity, J.P.A. orcid.org/0000-0001-5038-5699 (2022) A mild and regioselective route to fluoroalkyl aromatic compounds via directed cycloaddition reactions. The Journal of Organic Chemistry, 87 (15). pp. 9764-9768. ISSN 0022-3263
Cousins, D.L., Fricero, P., Kopf, K.P.M. et al. (4 more authors) (2021) Pyrimidin‐6‐yl trifluoroborate salts as versatile templates for heterocycle synthesis. Angewandte Chemie International Edition, 60 (17). pp. 9412-9415. ISSN 1433-7851
García-Vázquez, V., Hoteite, L., Lakeland, C.P. et al. (2 more authors) (2021) A Pd-catalyzed [4 + 2] annulation approach to fluorinated N-heterocycles. Organic Letters, 23 (7). pp. 2811-2815. ISSN 1523-7060
Zirimwabagabo, J.-O., Jailani, A.B.A. orcid.org/0000-0001-9837-6062, Avgoustou, P. orcid.org/0000-0002-1642-1083 et al. (10 more authors) (2021) Discovery of a first-in-class small molecule antagonist against the adrenomedullin-2 receptor: structure–activity relationships and optimization. Journal of Medicinal Chemistry, 64 (6). pp. 3299-3319. ISSN 0022-2623
Harrity, J.P.A. orcid.org/0000-0001-5038-5699, Mora-Radó, H., Czechtizky, W. et al. (1 more author) (2021) Design and synthesis of fused pyridine building blocks for automated library generation. ChemMedChem, 16 (2). pp. 328-334. ISSN 1860-7179
Harrity, J.P.A., Fricero, P., Bialy, L. et al. (2 more authors) (2020) Design and synthesis of novel pyrazole based heterotricycles and their derivatization via automated library synthesis. ChemMedChem, 15 (17). pp. 1634-1638. ISSN 1860-7179
Avgoustou, P., Jailani, A.B.A., Zirimwabagabo, J.-O. et al. (15 more authors) (2020) Discovery of a first-in-class potent small molecule antagonist against the adrenomedullin-2 receptor. ACS Pharmacology & Translational Science, 3 (4). pp. 706-719. ISSN 2575-9108
Al-Saedy, M.A.E. and Harrity, J.P.A. orcid.org/0000-0001-5038-5699 (2020) A practical and versatile method for the C–H sulfenylation of imidazo[1,2-a]pyridines. Synlett, 31 (12). pp. 1182-1184. ISSN 0936-5214
Holmes, T., Brown, A.W., Suggitt, M. et al. (5 more authors) (2020) The influence of hypoxia and energy depletion on the response of endothelial cells to the vascular disrupting agent combretastatin A-4-phosphate. Scientific Reports, 10 (1). 9926. ISSN 2045-2322
Harrity, J.P.A., Lakeland, C.P. and Watson, D.W. (2020) Exploiting synergistic catalysis for an ambient temperature photocycloaddition to pyrazoles. Chemistry – A European Journal, 26 (1). pp. 155-159. ISSN 0947-6539
Ball-Jones, M.P. orcid.org/0000-0001-9131-2373, Tyler, J., Mora-Radó, H. et al. (3 more authors) (2019) Exploiting hydrazones to improve the efficiency of 6π-electrocyclization reactions of 1-azatrienes. Organic Letters, 21 (17). pp. 6821-6824. ISSN 1523-7060
Brown, A.W., Holmes, T., Fisher, M. et al. (3 more authors) (2018) Cover feature : Evaluation of sydnone-based analogues of Combretastatin A-4 phosphate (CA4P) as vascular disrupting agents for use in cancer therapy (ChemMedChem 24/2018). ChemMedChem, 13 (24). p. 2600. ISSN 1860-7179
Harrity, J.P.A., Brown, A., Holmes, T. et al. (3 more authors) (2018) Evaluation of sydnone-based analogs of combretastatin A-4 phosphate (CA4P) as vascular disrupting agents for use in cancer therapy. ChemMedChem, 13 (24). pp. 2618-2626. ISSN 1860-7179
Harrity, J.P.A., Mora, H., Sotorrios, L. et al. (5 more authors) (2018) Synthetic and Mechanistic Investigation of an Oxime Ether Electrocyclization Approach to Heteroaromatic Boronic Acid Derivatives. Chemistry - A European Journal, 24 (38). pp. 9530-9534.
Maiden, T.M.M., Mbelesi, N., Procopiou, P.A. orcid.org/0000-0001-5907-116X et al. (2 more authors) (2018) A convergent strategy towards febrifugine and related compounds. Organic and Biomolecular Chemistry, 16 (22). pp. 4159-4169. ISSN 1477-0520
Kakaawla, T.K.K. and Harrity, J.P.A. orcid.org/0000-0001-5038-5699 (2018) Development of an amine-catalyzed regioselective synthesis of pyrroles. Organic Letters, 20 (1). pp. 201-203. ISSN 1523-7060
Fricero, P., Bialy, L., Czechtizky, W. et al. (2 more authors) (2018) Synthesis of bifunctional thiophenes via Fiesselmann condensation of ynone trifluoroborate salts. Organic Letters, 20 (1). pp. 198-200. ISSN 1523-7060
Al-Saedy, M.A.E., Nassoy, A.C.M.A. and Harrity, J.P.A. (2017) Accounting for different reactivities of sulfinate and thiosulfate salts in regioselective azetidine coupling via C–H sulfenylation of indoles. Synlett, 29 (03). pp. 349-353. ISSN 0936-5214
Allen, B.D.W., Lakeland, C.P. and Harrity, J.P.A. orcid.org/0000-0001-5038-5699 (2017) Frontispiece : Utilizing palladium-stabilized zwitterions for the construction of N-heterocycles. Chemistry - A European Journal, 23 (56). ISSN 0947-6539
Allen, B.D.W., Lakeland, C.P. and Harrity, J.P.A. (2017) Utilizing Palladium-Stabilized Zwitterions for the Construction of N-Heterocycles. Chemistry - A European Journal , 23 (56). pp. 13830-13857. ISSN 0947-6539
Brown, A.W. and Harrity, J.P.A. (2017) Expanding available pyrazole substitution patterns by sydnone cycloaddition reactions. Tetrahedron, 73 (22). pp. 3160-3172. ISSN 0040-4020
Harrity, J.P.A., Brown, A. and Comas-Barcelo, J. (2017) A Mild and Regiospecific Synthesis of Pyrazoleboranes. Chemistry - A European Journal , 23 (22). pp. 5228-5231. ISSN 0947-6539
Comas-Barceló, J. and Harrity, J.P.A. (2017) Metal Acetylides in Cycloaddition Reactions. Synthesis, 49 (06). pp. 1168-1181. ISSN 0039-7881
Allen, B.D.W., Connolly, M.J. and Harrity, J.P.A. (2016) Frontispiece: A Pd-Catalyzed Synthesis of Functionalized Piperidines. Chemistry - A European Journal, 22 (37). ISSN 0947-6539
Al-Saedy, M.A.E. and Harrity, J.P.A. (2016) Synthesis and Stabilities of 3-Borylated Indoles. Synlett, 27 (11). pp. 1674-1676. ISSN 0936-5214
Kakaawla, T.K.K., Hartley, W.C. and Harrity, J.P.A. (2016) Synthesis and Cycloaddition Reactions of Stabilized Münchnones. European Journal of Organic Chemistry, 2016 (16). pp. 2789-2792. ISSN 1434-193X
Mora-Radó, H., Bialy, L., Czechtizky, W. et al. (2 more authors) (2016) An alkyne diboration/6π-electrocyclization strategy for the synthesis of pyridine boronic acid derivatives. Angewandte Chemie, 128 (19). pp. 5928-5930. ISSN 0044-8249
Comas-Barceló, J., Blanco-Ania, D., van den Broek, S.A.M.W. et al. (3 more authors) (2016) Cu-catalysed pyrazole synthesis in continuous flow. Catalysis Science and Technology, 6 (13). pp. 4718-4723. ISSN 2044-4753
Edeson, S.J., Maduli, E.J.M., Swanson, S. et al. (2 more authors) (2016) Investigation of a Late-Stage Derivatization Approach to Isatogens: Discovery of New Reaction Pathways. European Journal of Organic Chemistry, 2016 (1). pp. 83-86. ISSN 1434-193X
Maiden, T.M.M., Swanson, S., Procopiou, P.A. et al. (1 more author) (2015) A Mild and Regioselective Route to Functionalized Quinazolines. Chemistry - A European Journal, 21 (41). pp. 14342-14346. ISSN 0947-6539
Nassoy, A-C.M.A., Raubo, P. and Harrity, J.P.A. (2015) Synthesis and indole coupling reactions of azetidine and oxetane sulfinate salts. Chemical Communications, 51 (27). 5914 - 5916. ISSN 1359-7345
Brown, A.W. and Harrity, J.P.A. (2015) Direct Arylation of Sydnones with Aryl Chlorides toward Highly Substituted Pyrazoles. Journal of Organic Chemistry , 80 (4). 2467 - 2472. ISSN 0022-3263
Comas-Barcelo, J., Foster, R.S., Fiser, B. et al. (2 more authors) (2015) Cu-Promoted Sydnone Cycloadditions of Alkynes: Scope and Mechanism Studies. Chemistry - A European Journal, 21 (8). 3257 - 3263. ISSN 0947-6539
Maduli, E.J.M., Edeson, S.J., Swanson, S. et al. (2 more authors) (2015) 2-Iodoisatogens: Versatile Intermediates for the Synthesis of Nitrogen Heterocycles. Organic Letters, 17 (2). 390 - 392. ISSN 1523-7060
Bachollet, S.P.J.T., Vivat, J.F., Cocker, D.C. et al. (2 more authors) (2014) Development of a Mild and Versatile Directed Cycloaddition Approach to Pyridines. Chemistry - A European Journal, 20 (40). 12889 - 12893. ISSN 0947-6539
Crepin, D.F.P., Harrity, J.P.A., Jiang, J. et al. (3 more authors) (2014) A Mechanistic Study of the Lewis Base-Directed Cycloaddition of 2-Pyrones and Alkynylboranes. Journal of the American Chemical Society, 136 (24). 8642 - 8653. ISSN 0002-7863
Edeson, S.J., Jiang, J., Swanson, S. et al. (4 more authors) (2014) Studies on the stereochemical assignment of 3-acylidene 2-oxindoles. Organic and Biomolecular Chemistry, 12 (20). 3201 - 3210. ISSN 1477-0520
Patent
The University of Sheffield (2018) WO2018211275 - COMPOUNDS. WO2018/211275Al.