Items where authors include "Overkleeft, Herman S."

Article

Pickles, Isabelle B., Chen, Yurong, Moroz, Olga et al. (9 more authors) (2024) Precision activity-based α-amylase probes for dissection and annotation of linear and branched-chain starch degrading enzymes. Angewandte Chemie International Edition. e202415219. ISSN 1433-7851

Koemans, Tony, Bennett, Megan, Ferraz, Maria J. et al. (6 more authors) (2024) Structure-Guided Design of C3-Branched Swainsonine as Potent and Selective Human Golgi α-Mannosidase (GMII) Inhibitor. Chemical Communications. ISSN 1364-548X

Artola, Marta, Aerts, Johannes M.F.G., van der Marel, Gijsbert A. et al. (4 more authors) (2024) From Mechanism-Based Retaining Glycosidase Inhibitors to Activity-Based Glycosidase Profiling. Journal of the American Chemical Society. pp. 24729-24741. ISSN 1520-5126

Su, Qin, Louwerse, Max, Lammers, Rob F. et al. (11 more authors) (2024) Selective labelling of GBA2 in cells with fluorescent β-d-arabinofuranosyl cyclitol aziridines. Chemical Science. pp. 15212-15220. ISSN 2041-6539

Thaler, Melissa, Ofman, Tim P., Kok, Ken et al. (16 more authors) (2024) Epi-cyclophellitol cyclosulfate, a mechanism-based ER α-glucosidase II inhibitor, blocks replication of SARS-CoV-2 and other coronaviruses. ACS Central Science. 1594–1608. ISSN 2374-7943 (In Press)

Borlandelli, Valentina, Offen, Wendy A orcid.org/0000-0002-2758-4531, Moroz, Olga et al. (9 more authors) (2023) β-L-Arabinofurano-cyclitol Aziridines are Cysteine-directed Broad-spectrum Inhibitors and Activity-based Probes for Retaining β-L-arabinofuranosidases. ACS Chemical Biology. 2564–2573. ISSN 1554-8937

McGregor, Nicholas George Sarre, De Boer, Casper, Foucart, Quentin Pierre Olivier et al. (6 more authors) (2023) A multiplexing activity-based protein profiling platform for dissection of a native bacterial xyloglucan-degrading system. ACS Central Science. pp. 2306-2314. ISSN 2374-7951

Males, Alexandra orcid.org/0000-0002-7250-8300, Kok, Ken, Nin-Hill, Alba et al. (8 more authors) (2023) Cyclosulfamidate Mannose-Configured Cyclitol Allows Specific Allele-Dependent Inhibition of GH47 α-D-Mannosidases Through a Bump-Hole Strategy. Chemical Science. pp. 13581-13586. ISSN 2041-6539

Su, Qin, Kuo, Ethan, van den Nieuwendijk, Rian et al. (12 more authors) (2023) The Development of a Broad-Spectrum Retaining β-Exo-Galactosidase Activity-Based Probe. Organic & biomolecular chemistry. 7813–7820. ISSN 1477-0539

van der Gracht, Daniël, Rowland, Rhianna J., Roig-Zamboni, Véronique et al. (7 more authors) (2023) Fluorescence Polarisation Activity-Based Protein Profiling in the Identification of Deoxynojirimycin-type Inhibitors selective for Lysosomal Retaining Alpha- and Beta-Glucosidases. Chemical Science. pp. 9136-9144. ISSN 2041-6539 (In Press)

Borlandelli, Valentina, Armstrong, Zachary, Nin-Hill, Alba et al. (6 more authors) (2023) 4-O-Substituted Glucuronic Cyclophellitols are Selective Mechanism-Based Heparanase Inhibitors. ChemMedChem. e202200580. ISSN 1860-7187

Kok, Ken, Kuo, Chi Lin, Katzy, Rebecca E. et al. (10 more authors) (2022) 1,6- epi-Cyclophellitol Cyclosulfamidate Is a Bona Fide Lysosomal α-Glucosidase Stabilizer for the Treatment of Pompe Disease. Journal of the American Chemical Society. 14819–14827. ISSN 1520-5126

Boer, Casper de, Armstrong, Zachary, Lit, Vincent A. J. et al. (15 more authors) (2022) Mechanism based heparanase inhibitors reduce cancer metastasis in vivo. Proceedings of the National Academy of Sciences of the United States of America. e2203167119. ISSN 1091-6490

McGregor, Nicholas G. S., Kuo, Chi-Lin, Beenakker, Thomas J. M. et al. (8 more authors) (2022) Synthesis of Broad-Specificity Activity-Based Probes for Exo-β-Mannosidases. Organic and Biomolecular Chemistry. pp. 877-886. ISSN 1477-0539

McGregor, Nicholas G.S., Boer, Casper de, Santos, Mikhaaeel et al. (6 more authors) (2022) Activity-Based Protein Profiling Reveals Dynamic Substrate-Specific Cellulase Secretion by Saprotrophic Basidiomycetes. Biotechnology for biofuels. 6. ISSN 1754-6834

Rowland, Rhianna J., Chen, Yurong, Breen, Imogen et al. (9 more authors) (2021) Design, Synthesis and Structural Analysis of Glucocerebrosidase Imaging Agents. Chemistry : A European Journal. ISSN 1521-3765

Schröder, Sybrin P., Offen, Wendy A. orcid.org/0000-0002-2758-4531, Males, Alexandra orcid.org/0000-0002-7250-8300 et al. (9 more authors) (2021) The development of non-hydrolysable oligosaccharide activity-based inactivators for endoglycanases:a case study on a-1,6 mannanases. Chemistry A European Journal. ISSN 1521-3765

McGregor, Nicholas G. S., Coines, Joan, Borlandelli, Valentina et al. (14 more authors) (2021) Cysteine Nucleophiles in Glycosidase Catalysis:Application of a Covalent β-L-Arabinofuranosidase Inhibitor. Angewandte Chemie International Edition. pp. 5754-5758. ISSN 1433-7851

Chen, Yurong, Armstrong, Zachary, Artola, Marta et al. (10 more authors) (2021) Activity-based protein profiling of retaining α-amylases in complex biological samples. Journal of the American Chemical Society. pp. 2423-2432. ISSN 1520-5126

McGregor, Nicholas G.S., Turkenburg, Johan P., Mørkeberg Krogh, Kristian B.R. et al. (5 more authors) (2020) Structure of a GH51 α- L -arabinofuranosidase from Meripilus giganteus:Conserved substrate recognition from bacteria to fungi. Acta Crystallographica Section D: Structural Biology. pp. 1124-1133. ISSN 2059-7983

De Boer, Casper, McGregor, Nicholas George Sarre, Peterse, Evert et al. (10 more authors) (2020) Glycosylated cyclophellitol-derived activity-based probes and inhibitors for cellulases. RSC Chemical Biology. pp. 148-155. ISSN 2633-0679

McGregor, Nicholas G.S., Artola, Marta, Nin-Hill, Alba et al. (12 more authors) (2020) Rational Design of Mechanism-Based Inhibitors and Activity-Based Probes for the Identification of Retaining α-l-Arabinofuranosidases. Journal of the American Chemical Society. pp. 4648-4662. ISSN 1520-5126

Jariwala, Parth B., Pellock, Samuel J., Cloer, Erica W. et al. (8 more authors) (2020) Discovering the Microbial Enzymes Driving Drug Toxicity with Activity-Based Protein Profiling. ACS Chemical Biology. pp. 217-225. ISSN 1554-8937

Wu, Liang orcid.org/0000-0003-0294-7065, Armstrong, Zach, Schröder, Sybrin P. et al. (5 more authors) (2019) An overview of activity-based probes for glycosidases. Current Opinion in Chemical Biology. pp. 25-36. ISSN 1367-5931

Artola, Marta, Hedberg, Christinne, Rowland, Rhianna J. et al. (11 more authors) (2019) α-D-Gal-cyclophellitol cyclosulfamidate is a Michaelis complex analog that stabilizes therapeutic lysosomal α-galactosidase A in Fabry disease. Chemical Science. ISSN 2041-6539

Schröder, Sybrin P., De Boer, Casper, McGregor, Nicholas G.S. et al. (22 more authors) (2019) Dynamic and Functional Profiling of Xylan-Degrading Enzymes in Aspergillus Secretomes Using Activity-Based Probes. ACS Central Science. pp. 1067-1078. ISSN 2374-7943

Artola, Marta, Kuo, Chi-Lin, Lelieveld, Lindsey T. et al. (7 more authors) (2019) Functionalized cyclophellitols are selective glucocerebrosidase inhibitors and induce a bona fide neuropathic Gaucher model in zebrafish. Journal of the American Chemical Society. 4214–4218. ISSN 1520-5126

Schröder, Sybrin P, Kallemeijn, Wouter W., Debets, Marjoke F et al. (10 more authors) (2018) Spiro-epoxyglycosides as Activity-Based Probes for Glycoside Hydrolase Family 99 Endomannosidase/Endomannanase. Chemistry : A European Journal. ISSN 1521-3765

Schröder, Sybrin P, Wu, Liang orcid.org/0000-0003-0294-7065, Artola, Marta et al. (9 more authors) (2018) Gluco-1 H-imidazole:A New Class of Azole-Type β-Glucosidase Inhibitor. Journal of the American Chemical Society. pp. 1-4. ISSN 1520-5126

Schroder, Sybrin P, van de Sande, Jasper W, Kallemeijn, Wouter W. et al. (13 more authors) (2017) Towards broad spectrum activity-based glycosidase probes: synthesis and evaluation of deoxygenated cyclophellitol aziridines. Chemical Communications. pp. 1-5. ISSN 1364-548X

Lahav, Daniël, Liu, Bing, van den Berg, Richard J. B. H. N. et al. (15 more authors) (2017) A Fluorescence Polarization Activity-Based Protein Profiling Assay in the Discovery of Potent, Selective Inhibitors for Human Nonlysosomal Glucosylceramidase. Journal of the American Chemical Society. pp. 14192-14197. ISSN 1520-5126

Wu, Liang orcid.org/0000-0003-0294-7065, Jiang, Jianbing, Jin, Yi orcid.org/0000-0002-6927-4371 et al. (12 more authors) (2017) Activity-based probes for functional interrogation of retaining β-glucuronidases. NATURE CHEMICAL BIOLOGY. pp. 867-873. ISSN 1552-4450

Artola, Marta, Wu, Liang orcid.org/0000-0003-0294-7065, Ferraz, Maria J. et al. (10 more authors) (2017) 1,6-Cyclophellitol Cyclosulfates:A New Class of Irreversible Glycosidase Inhibitor. ACS Central Science. pp. 784-793. ISSN 2374-7943

van Rijssel, Erwin, Janssen, Antonius P.A., Males, Alexandra orcid.org/0000-0002-7250-8300 et al. (4 more authors) (2017) Conformational behaviour of mannuronic acid based azasugars. Chembiochem. pp. 1-9. ISSN 1439-7633

Marques, André R. A., Willems, Lianne I. orcid.org/0000-0001-5411-1329, Herrera Moro, Daniela et al. (15 more authors) (2017) A Specific Activity-Based Probe to Monitor Family GH59 Galactosylceramidase, the Enzyme Deficient in Krabbe Disease. Chembiochem. pp. 402-412. ISSN 1439-7633

Beenakker, Thomas J. M., Wander, Dennis, Offen, Wendy A. orcid.org/0000-0002-2758-4531 et al. (13 more authors) (2017) Carba-Cyclophellitols are Neutral Retaining Glucosidase Inhibitors. Journal of the American Chemical Society. 6534–6537. ISSN 1520-5126