Brown, A.W. and Harrity, J.P.A. (2015) Direct Arylation of Sydnones with Aryl Chlorides toward Highly Substituted Pyrazoles. Journal of Organic Chemistry , 80 (4). 2467 - 2472. ISSN 0022-3263
Abstract
The direct arylation of the C4 position of both N-alkyl- and N-arylsydnones with aryl/heteroaryl chlorides has been realized. The reaction is quite general and allows access to a wide range of 4-substituted sydnones. Yields of more challenging substrates can be improved through the use of aryl bromides.
Metadata
Item Type: | Article |
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Authors/Creators: |
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Copyright, Publisher and Additional Information: | © 2015 American Chemical Society. This is an author produced version of a paper subsequently published in Journal of Organic Chemistry. Uploaded in accordance with the publisher's self-archiving policy. |
Dates: |
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Institution: | The University of Sheffield |
Academic Units: | The University of Sheffield > Faculty of Science (Sheffield) > Department of Chemistry (Sheffield) |
Depositing User: | Symplectic Sheffield |
Date Deposited: | 17 Aug 2015 15:42 |
Last Modified: | 09 Mar 2016 02:56 |
Published Version: | http://dx.doi.org/10.1021/acs.joc.5b00143 |
Status: | Published |
Publisher: | American Chemical Society |
Refereed: | Yes |
Identification Number: | 10.1021/acs.joc.5b00143 |
Related URLs: | |
Open Archives Initiative ID (OAI ID): | oai:eprints.whiterose.ac.uk:88792 |