Gorman, Ryan M., Hurst, Timothy E. orcid.org/0000-0003-0524-2909, Petersen, Wade F. et al. (1 more author) (2019) A copper(II)-mediated radical cross-dehydrogenative coupling/sulfinic acid elimination approach to 2-quinolones. Tetrahedron. 130711. ISSN 0040-4020
Abstract
A new cyclisation procedure to prepare 4-carboxy-quinolin-2-ones via a one-pot Cu(II)-mediated radical cross-dehydrogenative coupling/sulfinic acid elimination of linear anilides is described. Extensions to more complex substrates are also reported as are applications in target synthesis allowing access to natural products isolated from Oryza sativa and HOFQ.
Metadata
Item Type: | Article |
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Authors/Creators: |
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Copyright, Publisher and Additional Information: | © 2019 Elsevier Ltd. All rights reserved. This is an author-produced version of the published paper. Uploaded in accordance with the publisher’s self-archiving policy. |
Keywords: | 2-Quinolones,Cross-dehydrogenative coupling,Cu(II)-catalysis,Total synthesis |
Dates: |
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Institution: | The University of York |
Academic Units: | The University of York > Faculty of Sciences (York) > Chemistry (York) |
Depositing User: | Pure (York) |
Date Deposited: | 09 Dec 2019 10:50 |
Last Modified: | 16 Oct 2024 16:14 |
Published Version: | https://doi.org/10.1016/j.tet.2019.130711 |
Status: | Published online |
Refereed: | Yes |
Identification Number: | 10.1016/j.tet.2019.130711 |
Related URLs: | |
Open Archives Initiative ID (OAI ID): | oai:eprints.whiterose.ac.uk:154339 |
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