Discovery and Optimization of a Selective Ligand for the Switch/Sucrose Nonfermenting-Related Bromodomains of Polybromo Protein-1 by the Use of Virtual Screening and Hydration Analysis

Myrianthopoulos, V, Gaboriaud-Kolar, N, Tallant, C et al. (19 more authors) (2016) Discovery and Optimization of a Selective Ligand for the Switch/Sucrose Nonfermenting-Related Bromodomains of Polybromo Protein-1 by the Use of Virtual Screening and Hydration Analysis. Journal of Medicinal Chemistry, 59 (19). pp. 8787-8803. ISSN 0022-2623

Abstract

Metadata

Authors/Creators:
  • Myrianthopoulos, V
  • Gaboriaud-Kolar, N
  • Tallant, C
  • Hall, M-L
  • Grigoriou, S
  • Brownlee, PM
  • Fedorov, O
  • Rogers, C
  • Heidenreich, D
  • Wanior, M
  • Drosos, N
  • Mexia, N
  • Savitsky, P
  • Bagratuni, T
  • Kastritis, E
  • Terpos, E
  • Filippakopoulos, P
  • Müller, S
  • Skaltsounis, A-L
  • Downs, JA
  • Knapp, S
  • Mikros, E
Copyright, Publisher and Additional Information: © 2016 American Chemical Society. This is an open access article under the terms of the Creative Commons Attribution License (CC-BY 4.0), which permits unrestricted use, distribution and reproduction in any medium, provided the original work is properly cited. To view a copy of this license, visit http://creativecommons.org/licenses/by/4.0/.
Dates:
  • Published: 13 October 2016
  • Accepted: 12 September 2016
  • Published (online): 12 September 2016
Institution: The University of Leeds
Academic Units: The University of Leeds > Faculty of Arts, Humanities and Cultures (Leeds) > School of Design (Leeds)
Depositing User: Symplectic Publications
Date Deposited: 06 Mar 2019 16:01
Last Modified: 07 Mar 2019 13:46
Status: Published
Publisher: American Chemical Society
Identification Number: https://doi.org/10.1021/acs.jmedchem.6b00355

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