Picomolar, selective and subtype specific small-molecule inhibition of TRPC1/4/5 channels

Rubaiy, HN orcid.org/0000-0002-1489-5576, Ludlow, MJ, Henrot, M et al. (18 more authors) (2017) Picomolar, selective and subtype specific small-molecule inhibition of TRPC1/4/5 channels. Journal of Biological Chemistry, 292. pp. 8158-8173. ISSN 0021-9258

Abstract

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Authors/Creators:
Copyright, Publisher and Additional Information: © 2017, The American Society for Biochemistry and Molecular Biology. This is an open access article under the terms of the Creative Commons CC-BY license.
Keywords: calcium; calcium release-activated calcium channel protein 1 (ORAI1); ion channel; pharmacology; transient receptor potential channels (TRP channels); Englerin; Heteromeric channel; Non-selective cationic channel; Store-operated calcium entry; Transient Receptor Potential Canonical
Dates:
  • Published: 19 May 2017
  • Accepted: 21 March 2017
  • Published (online): 21 March 2017
Institution: The University of Leeds
Academic Units: The University of Leeds > Faculty of Maths and Physical Sciences (Leeds) > School of Chemistry (Leeds) > Organic Chemistry (Leeds)
The University of Leeds > Faculty of Medicine and Health (Leeds) > School of Medicine (Leeds) > Leeds Institute of Genetics, Health and Therapeutics (LIGHT) > Academic Unit of Cardiovascular Medicine (Leeds)
Depositing User: Symplectic Publications
Date Deposited: 23 Mar 2017 11:57
Last Modified: 27 Jan 2018 03:46
Published Version: https://doi.org/10.1074/jbc.M116.773556
Status: Published
Publisher: American Society for Biochemistry and Molecular Biology
Identification Number: https://doi.org/10.1074/jbc.M116.773556
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