Watson, EL, Ball, A, Raw, SA et al. (1 more author) (2016) Synthetic Studies on Psychotrimine: Palladium-Catalysed Arylation of 2-(N-Indolyl) Amides. SYNLETT, 27 (1). pp. 146-150. ISSN 0936-5214
Abstract
Through careful choice of conditions, 2-(N-indolyl) amides can be directed to undergo selectively either enolate arylation to give oxindoles or direct arylation to give indolo-fused benzodiazepines. The former chemistry facilitates the synthesis of the hexahydropyrrolindole core of psychotrimine.
Metadata
Item Type: | Article |
---|---|
Authors/Creators: |
|
Copyright, Publisher and Additional Information: | © 2015, Georg Thieme Verlag. This is an author produced version of a paper published in Synlett. Uploaded in accordance with the publisher's self-archiving policy. |
Keywords: | alkaloids - arylation - cyclisation - polycycles - total synthesis |
Dates: |
|
Institution: | The University of Leeds |
Academic Units: | The University of Leeds > Faculty of Engineering & Physical Sciences (Leeds) > School of Chemistry (Leeds) |
Depositing User: | Symplectic Publications |
Date Deposited: | 17 Nov 2015 16:35 |
Last Modified: | 16 Nov 2016 08:56 |
Published Version: | http://dx.doi.org/10.1055/s-0035-1560519 |
Status: | Published |
Publisher: | Georg Thieme Verlag |
Identification Number: | 10.1055/s-0035-1560519 |
Open Archives Initiative ID (OAI ID): | oai:eprints.whiterose.ac.uk:91920 |