Stapled Peptides as HIF‐1α/p300 Inhibitors: Helicity Enhancement in the Bound State Increases Inhibitory Potency

Hetherington, K, Hegedus, Z, Edwards, TA orcid.org/0000-0002-1467-3674 et al. (3 more authors) (2020) Stapled Peptides as HIF‐1α/p300 Inhibitors: Helicity Enhancement in the Bound State Increases Inhibitory Potency. Chemistry: A European Journal. ISSN 0947-6539

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Authors/Creators:
Copyright, Publisher and Additional Information: © 2020 The Authors. Published by Wiley-VCH Verlag GmbH & Co. KGaA. This is an open access article under the terms of the Creative Commons Attribution License, which permits use, distribution and reproduction in any medium, provided the original work is properly cited. To view a copy of this license, visit http://creativecommons.org/licenses/by/4.0/.
Keywords: chemical biology; oncology; peptidomimetics; protein–protein interactions; stapled peptides
Dates:
  • Accepted: 14 April 2020
  • Published (online): 19 April 2020
Institution: The University of Leeds
Academic Units: The University of Leeds > Faculty of Maths and Physical Sciences (Leeds) > School of Chemistry (Leeds) > Organic Chemistry (Leeds)
The University of Leeds > Faculty of Biological Sciences (Leeds) > School of Molecular and Cellular Biology (Leeds) > Crystallography (Leeds)
Depositing User: Symplectic Publications
Date Deposited: 17 Apr 2020 12:04
Last Modified: 08 Jun 2020 15:28
Status: Published online
Publisher: Wiley
Identification Number: https://doi.org/10.1002/chem.202000417

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