Items where authors include "McPhillie, MJ"

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Number of items: 16.

Article

Dokla, EME, Abutaleb, NS, Milik, SN orcid.org/0000-0001-6563-8265 et al. (9 more authors) (2023) SAR investigation and optimization of benzimidazole-based derivatives as antimicrobial agents against Gram-negative bacteria. European Journal of Medicinal Chemistry, 247. 115040. ISSN 0223-5234

Grossman, S, Fishwick, CWG and McPhillie, MJ orcid.org/0000-0001-8264-8211 (2023) Developments in Non-Intercalating Bacterial Topoisomerase Inhibitors: Allosteric and ATPase Inhibitors of DNA Gyrase and Topoisomerase IV. Pharmaceuticals, 16 (2). 261. ISSN 1424-8247

Orritt, KM, Feng, L, Newell, JF et al. (9 more authors) (2022) De novo design of type II topoisomerase inhibitors as potential antimicrobial agents targeting a novel binding region. RSC Medicinal Chemistry, 13 (7). pp. 831-839. ISSN 2632-8682

Turvey, SJ orcid.org/0000-0003-4298-8339, McPhillie, MJ orcid.org/0000-0001-8264-8211, Kearney, MT et al. (3 more authors) (2022) Recent Developments in the Structural Characterisation of the IR and IGF1R: Implications for the Design of IR-IGF1R Hybrid Receptor Modulators. RSC Medicinal Chemistry, 2022 (4). pp. 360-374. ISSN 2632-8682

M. E. Dokla, E, Kamal Abdel-Aziz, A, Milik, SN et al. (3 more authors) (2022) Discovery of a Benzimidazole-based Dual FLT3/TrKA Inhibitor Targeting Acute Myeloid Leukemia. Bioorganic and Medicinal Chemistry, 56. 116596. p. 116596. ISSN 0968-0896

Dokla, EME, Abdel-Aziz, AK, Milik, SN et al. (5 more authors) (2021) Indolin-2-one derivatives as selective Aurora B kinase inhibitors targeting breast cancer. Bioorganic Chemistry, 117. 105451. 105451-. ISSN 0045-2068

Orritt, KM, Maxwell, A, Fishwick, CWG orcid.org/0000-0003-1283-2181 et al. (1 more author) (2021) Exploitation of a novel allosteric binding region in DNA gyrase and its implications for antibacterial drug discovery. Future Medicinal Chemistry. ISSN 1756-8919

Pavić, A, Ji, Y, Serafini, A et al. (8 more authors) (2020) Functional Characterization of the γ-Aminobutyric Acid Transporter from Mycobacterium smegmatis MC2 155 Reveals Sodium-Driven GABA Transport. Journal of Bacteriology. ISSN 0021-9193

Shimizu, JF, Martins, DOS, McPhillie, MJ orcid.org/0000-0001-8264-8211 et al. (5 more authors) (2020) Is the ADP ribose site of the Chikungunya virus NSP3 Macro domain a target for antiviral approaches? Acta Tropica, 207. 105490. p. 105490. ISSN 0001-706X

McPhillie, MJ orcid.org/0000-0001-8264-8211, Zhou, Y, Hickman, MR et al. (31 more authors) (2020) Potent Tetrahydroquinolone Eliminates Apicomplexan Parasites. Frontiers in Cellular and Infection Microbiology, 10. 203. ISSN 2235-2988

Chandrabalan, A, McPhillie, MJ orcid.org/0000-0001-8264-8211, Morice, AH et al. (2 more authors) (2019) N-cinnamoylanthranilates as human TRPA1 modulators: Structure-activity relationships and channel binding sites. European Journal of Medicinal Chemistry, 170. pp. 141-156. ISSN 0223-5234

El Bissati, K, Redel, H, Ting, L-M et al. (7 more authors) (2019) Novel Synthetic Polyamines Have Potent Antimalarial Activities in vitro and in vivo by Decreasing Intracellular Spermidine and Spermine Concentrations. Frontiers in Cellular and Infection Microbiology, 9. 9. ISSN 2235-2988

lykins, JD, Filippova, E, Halavaty, AS et al. (21 more authors) (2018) CSGID Identifies Phenotypes and Solves Structures for Five Enzymes in Toxoplasma gondii. Frontiers in cellular and infection microbiology, 8. ARTN352. ISSN 2235-2988

Rawson, S orcid.org/0000-0002-2973-2630, Bisson, C, Hurdiss, DL et al. (6 more authors) (2018) Elucidating the structural basis for differing enzyme inhibitor potency by cryo-EM. Proceedings of the National Academy of Sciences of the United States of America, 115 (8). pp. 1795-1800. ISSN 0027-8424

Rawson, S, McPhillie, MJ, Johnson, RM et al. (2 more authors) (2017) The potential use of single-particle electron microscopy as a tool for structure-based inhibitor design. Acta Crystallographica Section D: Structural Biology, 73 (6). pp. 534-540. ISSN 2059-7983

Gordon, JA, Fishwick, CW orcid.org/0000-0003-1283-2181 and McPhillie, MJ (2017) New Opportunities in the Structure-based Design of Anti-Protozoan Agents. Current Topics in Medicinal Chemistry, 17 (1). pp. 79-90. ISSN 1568-0266

This list was generated on Sun Mar 24 08:02:21 2024 GMT.